Novel phenylamino acetamide derivatives as potent and selective κ opioid receptor agonists

Guo Hua Chu, Minghua Gu, Joel A. Cassel, Serge Belanger, Gabriel J. Stabley, Robert N. DeHaven, Nathalie Conway-James, Mike Koblish, Patrick J. Little, Diane L. DeHaven-Hudkins, Roland E. Dolle

Research output: Contribution to journalArticle

7 Scopus citations

Abstract

A novel series of phenylamino acetamide derivatives was synthesized. These amides were shown to be potent and selective κ opioid receptor agonists.

Original languageEnglish
Pages (from-to)645-648
Number of pages4
JournalBioorganic and Medicinal Chemistry Letters
Volume16
Issue number3
DOIs
StatePublished - Feb 1 2006
Externally publishedYes

Keywords

  • Analgesic
  • κ Opioid-receptor agonists

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  • Cite this

    Chu, G. H., Gu, M., Cassel, J. A., Belanger, S., Stabley, G. J., DeHaven, R. N., Conway-James, N., Koblish, M., Little, P. J., DeHaven-Hudkins, D. L., & Dolle, R. E. (2006). Novel phenylamino acetamide derivatives as potent and selective κ opioid receptor agonists. Bioorganic and Medicinal Chemistry Letters, 16(3), 645-648. https://doi.org/10.1016/j.bmcl.2005.10.034