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Differential megakaryocytic desensitization to platelet agonists
G. W. Dorn
, M. G. Davis
Roy and Diana Vagelos Division of Biology & Biomedical Sciences (DBBS)
Institute of Clinical and Translational Sciences (ICTS)
Department of Medicine
Division of Pharmacogenomics
DBBS - Molecular Cell Biology
DBBS - Human and Statistical Genetics
DBBS - Molecular Genetics and Genomics
Research output
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Contribution to journal
›
Article
›
peer-review
22
Scopus citations
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Keyphrases
Desensitization
100%
Platelets
100%
Megakaryocytic
100%
Platelet Agonists
100%
Protein Kinase
75%
Thrombin
75%
Phospholipase C
50%
Calcium Signaling
50%
Thromboxane A2 (TXA2)
50%
Megakaryocytes
50%
Platelet-activating Factor
50%
U46619
50%
Hydrolysis
25%
Bone Marrow
25%
Effective Concentration
25%
Staurosporine
25%
Phosphatidylinositol
25%
Phorbol 12-myristate 13-acetate
25%
Pharmacological Inhibitors
25%
Human Platelets
25%
Cytosolic Calcium
25%
Peripheral Circulation
25%
Calcium Response
25%
Calcium Desensitization
25%
Cell Inhibition
25%
Calcium Transient
25%
Inositol
25%
Fura-2
25%
Platelet-activating Factor Receptor
25%
Heterologous Desensitization
25%
Concentration Value
25%
Homologous Desensitization
25%
Dienoic Acids
25%
Protein Kinase C Activation
25%
Pharmacology, Toxicology and Pharmaceutical Science
Desensitization
100%
Protein Kinase C
80%
Thrombin
60%
Thromboxane A2
40%
15 Hydroxy 11alpha,9alpha Epoxymethanoprosta 5,13 Dienoic Acid
40%
Thrombocyte Activating Factor
40%
Lecithinase
40%
Staurosporine
20%
Phosphatidylinositol
20%
12-O-Tetradecanoylphorbol-13-Acetate
20%
Inositol
20%
Thrombocyte Activating Factor Receptor
20%
Fura-2
20%
EC50
20%